1-[(1S)-(4-Fluorophenyl)-((1′S)-1′-naphthalen-1-yl-ethylamino)-methyl]-naphthalen-2-trifluoromethanesulfonate
نویسندگان
چکیده
The complex structure of aminobenzylnaphthols can be easily obtained with the useful Betti reaction. These valuable compounds give rise to chiral intermediates, that found wide application in asymmetric synthesis. 1-[(1S)-(4-Fluorophenyl)-((1′S)-1′-naphthalen-1-yl-ethylamino)-methyl]-naphthalen-2-ol 1 was treated triflic anhydride yield corresponding (S,S)-triflate 2, which is a intermediate future synthesis aminophosphine, used catalysis. Preliminarily structural considerations based upon H(1)-NMR spectroscopy are also reported.
منابع مشابه
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ژورنال
عنوان ژورنال: Molbank
سال: 2023
ISSN: ['1422-8599']
DOI: https://doi.org/10.3390/m1695